1. Alvaro G. Temprano, Beatriz Sanchez de Blas, Concepción Pérez-Melero, Ricardo Espinosa-Escudero, Oscar Briz, Paula Cinca-Fernando, Lucia Llera, Maria J. Monte, Francisco A. Bermejo-Gonzalez, Jose J.G. Marin and Marta R. Romero.
Synthesis, characterization, and potential usefulness in liver function assessment of novel bile acid derivatives with near-infrared fluorescence (NIRBAD)
Bioconjugate Chem. 2024, DOI 0.1021/acs.bioconjchem.4c00168
2. Elena González-Hernández, Rubén Aparicio, Mercedes Garayoa, M. José Montero, M. Ángeles Sevilla and Concepción Pérez-Melero.
Dihydropyrimidine-2-thiones as Eg5 inhibitors and L-type calcium channel blockers: potential antitumour dual agents
Med. Chem. Commun. 2019, 10, 1589-1598
3. Concepción Pérez-Melero.
KSP inhibitors as antimitotic agents
Current Topics in Medicinal Chemistry2014, 14, 2286-2311
4. Concepción Álvarez, Raquel Álvarez, Purificación Corchete, Concepción Pérez-Melero, Rafael Pelaez and Manuel Medarde.
Exploring the effect of 2,3,4-trimethoxyphenyl moiety as a component of indolephenstatins
European Journal of Medicinal Chemistry 2010, 45, 588-597
5. Concepción Álvarez, Raquel Álvarez, Purificación Corchete, Concepción Pérez-Melero, Rafael Pelaez and Manuel Medarde.
Naphthylphenstatins as tubulin ligands: synthesis and biological evaluation
Bioorganic and Medicinal Chemistry 2008, 16, 8999-9008
6. Concepción Álvarez, Raquel Álvarez, Purificación Corchete, José Luis López, Concepción Pérez-Melero, Rafael Pelaez and Manuel Medarde.
Diarylmethyloxime and hydrazone derivatives with 5-indolyl moieties as potent inhibitors of tubulin polymerization
Bioorganic and Medicinal Chemistry 2008, 16, 5952-5961
7. Carmen Mateo, Raquel Álvarez, Concepción Pérez-Melero, Rafael Peláez and Manuel Medarde.
Conformationally restricted macrocyclic analogues of combretastatins
Bioorganic and Medicinal Chemistry Letters 2007, 17, 6316-6320
8. Concepción Álvarez, Raquel Álvarez, Purificación Corchete, Concepción Pérez-Melero, Rafael Peláez and Manuel Medarde.
Synthesis and biological activity of naphthalene analogues of phenstatins: Naphthylphenstatins
Bioorganic and Medicinal Chemistry Letters 2007, 17, 3417-3420
9. Carmen Mateo, Concepción Pérez-Melero, Rafael Peláez and Manuel Medarde.
Synthesis of a conformationally restricted polyoxygenated crownophane
Tetrahedron Letters 2005, 46 (41), 7055-7057
10. Finian Leeper, Dan Hawksley, Stéphane Mann, Concepción Pérez-Melero and Martin D. H. Wood.
Studies on thiamine diphosphate-dependent enzymes
Biochemical Society Transactions 2005, 33, 772-775
11. Carmen Mateo, Concepción Pérez-Melero, Rafael Peláez and Manuel Medarde.
Stilbenophane analogues of deoxycombretastatin A-4
Journal of Organic Chemistry 2005, 70, 6544-6547
12. Ana B. S. Maya, Concepción Pérez-Melero, Carmen Mateo, Dulce Alonso, José Luis Fernández, Consuelo Gajate, Faustino Mollinedo, Rafael Peláez, Esther Caballero and Manuel Medarde.
Further naphthylcombretastatins. An investigation on the role of the naphthalene moiety
Journal of Medicinal Chemistry 2005, 48 (2), 556-568
13. Ana B. S. Maya, Concepción Pérez-Melero, Rafael Peláez, Esther Caballero and Manuel Medarde.
New naphthylcombretastatins. Modifications on the ethylene bridge
Bioorganic and Medicinal Chemistry 2005, 13 (6), 2097-2107
14. Concepción Pérez-Melero, Ana B. S. Maya, Benedicto del Rey, Rafael Peláez, Esther Caballero and Manuel Medarde.
A new family of quinoline and quinoxaline analogues of combretastatins
Bioorganic and Medicinal Chemistry Letters 2004, 14, 3771-3774
15. Manuel Medarde, Ana B. S. Maya and Concepción Pérez-Melero.
Naphthalene combretastatin analogues. Synthesis, cytotoxicity and antitubulin activity
Journal of Enzyme Inhibition and Medicinal Chemistry 2004, 19 (6), 521-540
16. Stéphane Mann, Concepción Pérez-Melero and Finian J. Leeper.
Inhibition of thiamin diphosphate dependent enzymes by 3-deazathiamin diphosphate
Organic and Biomolecular Chemistry 2004, 2, 1732-1741
17. Luis G. Sevillano, Concepción P. Melero, Esther Caballero, Fernando Tomé, Lionel G. Lelièvre, Kathi Geering, Gilles Crambert, Rosalía Carrón, Manuel Medarde y Arturo San Feliciano.
Inotropic activity of hydroindenic amidinohydrazones
Journal of Medicinal Chemistry 2002, 45, 127-136
18. Concepción P. Melero, Manuel Medarde and Arturo San Feliciano.
A short review on cardiotonic steroids and their aminoguanidine analogues
Molecules 2000, 5, 51-81
19. Luis G. Sevillano, Concepción P. Melero, Melchor Boya, José Luis López, Fernando Tomé, Esther Caballero, Rosalía Carrón, M. José Montero, Manuel Medarde and Arturo San Feliciano.
Synthesis and inotropic activity of hydroindene derivatives
Bioorganic and Medicinal Chemistry 1999, 7, 2991-3001
20. Concepción P. Melero, Luis G. Sevillano, Esther Caballero, Fernando Tomé, Rosalía Carrón, M. José Montero, Arturo San Feliciano and Manuel Medarde.
Hydroindenic guanylhydrazones. Synthesis and evaluation as inotropic agents
Bioorganic and Medicinal Chemistry Letters 1998, 8, 3217-3222
21. Manuel Medarde, Esther Caballero, Concepción P. Melero, Fernando Tomé and Arturo San Feliciano.
Asymmetric synthesis of (+)-3a-Hydroxy-4,7a-dimethylperhydroindane-1,5-dione
Tetrahedron Asymmetry 1997, 8 (13), 2075-2077
22. Manuel Medarde, Esther Caballero, Fernando Tomé, Concepción P. Melero, Melchor Boya y Arturo San Feliciano.
Análogos sintéticos de cardenolidas con estructura simplificada. Derivados perhidroindénicos
Anales de Química 1995, 91, 89-94
23. Manuel Medarde, Fernando Tomé, José Luis López, Esther Caballero, Melchor Boya, Concepción P. Melero and Arturo San Feliciano.
Stereochemical control of perhydroindenes for the synthesis of cardenolide analogues
Tetrahedron Letters 1994, 35, 8683-8686
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